A-C
A-C | D-L | M-P | S-Z
Aldactone
Aldactone is a
diuretic and belongs to the subgroup of potassium-sparing
diuretics. Aldactone is an aldosterone antagonist. It
influences the body's own hormone, aldosterone, which
accelerates the excretion of potassium and reduces the
excretion of sodium and water Simplified; aldosterone
regulates the endogenous water household. The higher the
aldosterone level, the more water is stored in the body.
The use of Aldactone results in a significant reduction
in the aldosterone level so that an increased excretion
of sodium and water occurs while, at the same time,
potassium is reabsorbed. This also explains why Aldactone
is called a potassium-sparing diuretic since it does not
cause a loss of potassium like thiazides and furosemides.
Athletes must strictly observe that during the use of
Aldactone no additional potassium is taken since this
would cause a life-threatening increase in the serum
potassium level. Potassium sparing diuretics have
relatively low diuretic effects so that Aldactone can be
called a mild diuretic. It is interesting to note that
Aldactone is also an antiandrogen since it reduces the
androgen level. Female athletes take advantage of this
characteristic by using it to minimize the virilization
symptoms during steroid treatment or the symptoms after
treatment. For this purpose Aldactone is normally taken
daily for 10 to 14 days, usually in a dose of 50 mg/day.
In men this could cause problems since the relationship
of the androgen level to the estrogen level changes in
favor of the latter Thus, common side effects in men
include pain in the nipples and breast swelling (gynecomastia).
Bodybuilders use Aldactone almost exclusively during the
last week before a competition. Since this causes neither
a dramatic nor an immediately noticeable draining effect,
it is usually taken over 5-6 days in a dosage of 2
tablets of 50 mg daily. Aldactone should not be used to
expediently drain water at the last minute. Both male and
female athletes take it. The side effects of potassium-saving
diuretics are relatively low compared to thiazides and
furosemides. The main problems in men consist of
gynecomastia and possible impotence. Other side effects
can be low blood pressure, muscle spasms, dizziness,
gastrointestinal pain, vomiting, irregular pulse rate,
and fatigue. It is important to note that there is Ii',
significant increase in the serum potassium level (see
above).
Aldactone is a prescription drug available in American
pharmacies. Aldactone by Hoehringer Mannheim of Germany
is often found on be black market. A package contains 50
degrees of 50 mg each and costs approx. $30. On the black
market. The Mexican Aldactone by Searle can also
frequently be found on the black market. The 25-mg
tablets are of light-brown color; indented, and have a
SEARLE imprint. The original package contains three
strips, each with 10 tab-lets. There are currently no
Aldactone fakes available.
Anadrol
Anadrol was the U.S.
brand name for 50mg Oxymetholone tablets, which were
available in the U.S. until 1993. Syntex is the world
producer of this drug, and markets it under a few
different brand names in other areas. Oxymetholone is a
17alpha alkylated oral steroid. Second to none, this
product is generally considered the most powerful steroid
available. Anadrol will produce extremely dramatic weight
and strength gains in its user. Some of this weight and
strength gain will be due to the drugs heavy water
retention. Users of Anadrol report severe crashes when
stopping usage, mostly due to the loss of water and
inhibited endogenous hormone production brought about
during the cycle. Aside from the water, Anadrol will pack
on the mass like no other steroid. A short cycle of
Anadrol could account for a gain of over 20lbs in many
users, sometimes more. As this drugs anabolic properties
are so extreme, so are it's androgenic side effects. Due
to the strength of these side effects, Anadrol should
never be used by women. For starters, oxymetholone will
easily convert to estrogen and DHT. As stated earlier
water retention will be present, along with an increase
in blood pressure. Kidney functions may also need to be
looked after during longer use. Hair loss has also been
reported among users with a predisposition for male-pattern
baldness. The most dangerous attribute of Anadrol is that
is it 17alpha alkylated. As you probably know 17aa orals
are toxic to the liver. Unlike Dianabol (another popular
17aa oral) which is effective in doses of as little as 15mg,
Anadrol users generally start with 50mg/day and often
lead up to 150mg/day. So when a user takes 3 Anadrol
tablets, his liver is processing roughly the equivalent
of 30 Dianabol tablets. This obviously is quite a lot of
17aa steroid for your liver to process, so it is
pertinent a user has his liver enzymes checked regularly
with a doctor. When you hear of horror stories involving
liver cancer from steroid use, Anadrol is most often the
culprit. For medical treatment, Syntex recommends 1-5mg/kg
of bodyweight per day. This leads many patients to take
as many as 8+ tabs per day, for extended periods of time.
This is much more than an athlete would need and should
be using, which may be why documented cases of liver
cancer seem more prominent among non-athletes taking
Anadrol medically. Lately, many people are speculating on
how long this product will be available worldwide. Syntex
has stopped production of Anadrol in the U.S., Oxitosona
in Spain and medical use in other areas of the world
seems to be declining due to the advent of newer drugs to
treat conditions in which Anadrol was formerly used.
Aside from the Mexican version, all other forms of
Anadrol are now being counterfeited, often with
incredible accuracy. In the U.S., a version of the now
unavailable American Anadrol has been found in which box,
bottle and even the stamping of the tablet are identical
to the real version. The only seen difference is the lack
of active ingredient. Since real U.S. Anadrol has been
out of production for some time, it would be safe to say
anything labeled Anadrol is fake. Anapolon is copied as
well with good accuracy. Oxitosona was/is counterfeited
but since Syntex dropped its production in 1993, all
forms should be considered fake. Hemogenin from Brazil is
another popular version, which makes its way to the
states and is also counterfeited. Currently, all the
loose red Anadrols from Mexico (Stamped with SYNTEX on
one side and 2902 on the other) which are circulating the
states should be considered real. They are available only
to clinics and hospitals in Mexico, so black market
supplies are limited. Reports are that they may also be
slightly underdosed.
Anavar
(oxandrolone)
2.5mg tab 100/bottle Also under the name Lipo-Dex and
Nilavar.
Anavar
is manufactured by searle lavatories under the brand
name, and by spa labs under the generic name Oxandrolone.
The brand name drug is made under a certain number of
loss per year. This if it sells out before the end of the
year, the product just disappears. Searle does not make
more until the next term. This keeps the price of anavar
high, and availability low. Anavar is typically
prescribed on a 2 - tablet, twice daily routine. The drug
is better absorbed when taken right after meals. Woman
have started with one tablet twice daily. This is thought
to be the optimal dose for woman. The drug can be used in
combination with other steroids for optimum results after
a plateau is reached on the anavar alone. If some size is
required, but no injection is desired, dianabol or
anadrol can be combined with the anavar. Here the user
would add 1 dianabol tab twice daily or a half anadrol
twice daily. Later, and for greater size, going to 4
dianabol tabs, or to anadrol per day has worked well .
for greater gains the user would add an injectable
steroid to the cycle instead of the previously mentioned
orals. The injection would vary from deca for cutting, to
testosterone for weight and strength gains. Research
shows that anavar is the one anabolic steroid least
likely to cause any side effects . there are very rarely
reports of ill effects of any kind using anavar . there
is seldom any fluid gains with this drug, which makes it
the drug of choice with potential blood pressure problem
uses . anavar is also good trade for persons who need to
keep their weight down, either for cutting or like a
powerlifter who needs to make weight . Thus you will see
a number of bodybuilders using anavar the last two months
before competing. Some powerlifters claim that this
steroid is No. 1 for gaining strength without water
weight. The use of the low androgenic product is quite
popular with women. Very little masculinisation in any
form have been seen among woman who have used this trade
at a dose of 5 mg daily. Most women start out on 1 tablet
per day and go up to three tablets daily. The dosage of 5
mg of anavar per day has worked out to be the optimum.
The first signs of virilisaton could include persistent
hoarseness, deepening of the women's voice, acne,
decreased libido, and/or clitoral enlargement. If any of
these symptoms should show, the woman should get of the
trade immediately. Anavar will not aromatize. This means
of course it's one of the very few anabolic steroids that
will not convert to estrogen at any dosage. This means it
will not cause that soft look to the muscles or will it
lead to the development of breast tissue in men. Some
persons will convert much more of a steroid to estrogen
than others. These people can use a dosage starting with
2 tabs twice daily, and reaching a maximum dose of .1 MG
of the add per pound of body weight. Often the user
plateaus on the drug alone, he might add a small dose of
deca that would not aggravate any existing gynecomastia.
Or a daily dose of 10 MG of halotestin could be added to
the anavar cycle to increase strength and hardness, while
having no aromatize in effect. Anavar is a multi-purpose
steroid. Its very low toxicity makes it safe to take,
even on lower cycles. It is advised that a high protein
diet be maintained while taking anavar to insure its
effectiveness. It is been counterfeit under the Spa label.
Watch for the Searle liable to be safe.
Andriol
(Androxon,
Undestor, Restandol)
Introduction
There are two issues in relation to Andriol. First, there
exists a mythology that Andriol is totally useless.
Second, many who purchase Andriol have been grossly
misled. This article debunks the myth and offers some
solace to the misled. Many condemn Andriol through lack
of knowledge without considering that, since WAR and
others, including the medical community in most
countries, regard Andriol as effective, then perhaps it
has its uses. This misguided condemnation leads those who
should be considering Andriol to ignore it. On the other
hand, the over-enthusiastic words of some writers in
respect of Andriol have misled many novice Body Builders
(BB) to purchase Andriol when in fact it is unlikely to
be the most appropriate Anabolic Steroid (AS) for them.
Unthinking condemnation is particularly unwarranted given
that the principal agent in the ever popular Sustanon 250
(ie 100mg testosterone decanoate) is chemically identical
to the Testosterone Undecanoate (TU) in Andriol. Indeed,
chemically and mathematically, 1 bottle of Andriol is
equivalent to 24 Sustanon, but in practical application
and effectiveness they are poles apart. However, there
are a variety of problems associated with the use of
Andriol, not least of which is the fact that many
capsules purchased by BB are probably inert by the time
they are purchased. The problems associated with Andriol
and its potential for use by BB are examined below.
Description
Andriol (also know as Restandol, Undestor, Virigen,
Androxon and Panteston) is an oral testosterone androgen
compound whose prime agent is testosterone undecanoate (TU).
Andriol is supplied, by its sole manufacturer Organon, as
an oval, reddish-brown, soft gelatine capsule, marked
"ORG" and "D3V", containing 40mg of
TU in oleic acid. The capsule's non-medicinal ingredients
are: gelatine, glycerol, iron oxide red (E172), karion 83,
sodium ethyl hydroxybenzoate, sodium propyl
hydroxybenzoate and titanium dioxide. Andriol is supplied
in of bottles of 28, 56, 60 and 100 capsules dependent
upon country of manufacture. It is also supplied in foil
strips in Brazil and Thailand.
Pharmacology (per Rxmed)
Testosterone Undecanoate, an orally active testosterone
preparation, is a fatty acid ester of the natural
androgen testosterone. Unlike other oral testosterone
preparations, TU is able to by-pass the liver via the
lymphatic system and is therefore orally bioavailable.
Therapy with Andriol increases plasma levels of
testosterone and its active metabolites, leading to a
regular therapeutic effect. In eugonadal men, peak
testosterone levels are reached in approximately 4 to 5
hours after ingestion returning to basal levels after
about 10 hours. In volunteers and hypogonadal (ie. low
natural testosterone) men, 77 to 93% of an orally
administered dose of TU was excreted in the urine and
faeces within 3 to 4 days.
Storage is Critical
It is probably true to say that some of the Andriol
available on the Black Market is useless and serves no
purpose other than as a laxative. The reason is that,
unless refrigerated, Andriol will become inert after 3
months storage at room temperature (ie up to 30 degrees C).
Indeed, some claim that, at room temperature, it will
become inert after 2 months. Prolonged storage at higher
than room temperatures will clearly shorten this period.
Exposure to high temperatures will also cause the
capsules to become misshapen and even to melt. The
capsules should be stored in a refrigerator at a
temperature between 2 - 8 degrees C. Ideally, the bottle
of capsules should be removed from the refrigerator about
24 hrs before use, and once in use, the bottle should not
be returned to the refrigerator ie it should only be
ingested when fully thawed out.
The Problem
The problem with Andriol is that it is very idiosyncratic.
It does nothing for some, but for others it works for a
variety of purposes. This idiosyncratic feature reflects
both Andriol's delivery method and the nature of
individual metabolisms. Research has shown that, for some
people, only 3% - 4% of the Andriol ingested survives to
perform a useful function - for others the percentage is
higher, but never 100%. It is possible that, for most
people, less than 10% of the TU ingested survives to
become bioavailable. Another problem associated with
Andriol has been outlined by Dan Duchaine, who has
suggested that, of the small percentage of Andriol that
survives its journey through the gut to reach the
lymphatic system, 70% is converted into DHT. The
potential ramifications of DHT in the context of hair
loss and prostate are well known to all BB. However, the
amount of DHT arising from normal doses of Andriol is
unlikely to be significant, given the small percentage
that survives ingestion. Nevertheless this may account
for the anecdotal, but unsubstantiated, claims of Andriol
encouraging male-pattern baldness. Even for those for
whom Andriol does work, it takes trial and error over
time to establish a viable dose amount & schedule.
This dosage methodology is time consuming and expensive,
and although feasible in the medical environment, it is
less so in BB. The variability of Andriol's effectiveness
partly explains why 'Animal' on Varix states that Andriol
works and points to the overwhelming medical research
supporting it, while Human..saurus-rex on Anabolex says
to forget the medical evidence and that it does not work
for BB. Both are correct: statistically, medically,
chemically, scientifically, etc, Andriol does work, but
often not in a manner that is useful for young, healthy
BB.
Its Strong Points
Andriol's real strong point is in medical applications.
For instance, the efficacy of Andriol for use in androgen
replacement has been established in so many studies that
it is beyond dispute. Similarly Andriol's lack of
toxicity and safety in long term use (up to 10 yrs) has
also been clearly established.
Andriol is perhaps best suited for those BB who:
1. have a definite medical need e.g. liver function
problems, depression, thyroid problems, low natural
testosterone, other hormonal imbalances, osteoporosis;
infertility or
2. are aged over (say) 35 and thus have declining natural
testosterone levels. There are those who advocate that
the majority of men over 40 should adopt a regular
androgen supplementation regime using a mild form of
testosterone such as Andriol; and possibly for
3. 'hobby' BB who are more concerned with extreme safety
and are less concerned with quick results and expense.
Except for the above, Andriol is simply not cost-effective
relative to the other relatively safe options available e.g.
primobolan-depot.
There does appear to be a correlation between Andriol's
anecdotal effectiveness and age - older BB consider it
more useful than younger BB. This reflects the natural
age-related decline in testosterone. This decline is, at
its extreme, represented by the medical condition of
hypogonadism, for which one of the popular treatments
outside the USA is Andriol. For age-related male
testosterone deficiency which has not fallen to the level
of hypogonadism, namely the "viropause" or
"andropause", again Andriol, or alternatively
the testosterone patch, is the treatment of choice of
endocrinologists in many countries. In this area of low
normal and sub-normal natural testosterone levels,
Andriol is especially useful for the older BB.
Testosterone Undecanoate in injectable form, although not
generally available, is far less idiosyncratic than the
capsules. Indeed there is strong evidence to show that
injected TU is far superior to, for example, testosterone
enanthate. TU cream also has its uses, for example, it
has been shown to stimulate the growth of female pubic
hair. It has also been shown Andriol, taken in
conjunction with Nolvadex (tamoxifen citrate) can
significantly improve male fertility.
One of the most interesting things about TU (in either
form) is that it causes a significant decrease in the
level of Sex Hormone Binding Globulin (SHBG) which for
most males (incl. BB) is to the good. For example, in one
well-known study SHBG was reduced from 73.9 nmol/L to 35.1
at 3 months and to 29.2 at 6 months. Since SHBG
interferes with the bioavailability of testosterone (ie
it reduces "free T") and, perhaps, other
steroids, this leads to the speculation that perhaps TU
could be used in combination with other more anabolic
steroids as a synergist. It is debatable whether Andriol
is a useful general treatment in relation to AIDS, but
this reflects the multi-faceted nature of AIDS rather an
adverse comment on Andriol. There are some indications
that Andriol may be useful in assisting to normalise the
testosterone levels of AIDS sufferers. Current medical
guidelines for the normalisation of serum testosterone in
HIV suffers recommends 3 - 4 capsules (ie 120 - 160mg)
per day as an alternative to treatment with 200 - 400mg
of testosterone enanthate every 4 weeks.
How To Use It If You're Stuck With It
The foregoing does not assist the typical healthy BB who
might already have purchased Andriol. In such a
situation, 5 options appear open:
1. Use for Depression
Depression is an area where the average BB might find
Andriol useful. It has been shown from the work done on
hypogonadal men that (subject to dose) Andriol relieves,
and indeed can eliminate, the depression induced by low
serum T levels. Given that many BB suffer, among other
things, from depression and low natural testosterone
level when coming off a heavy AS cycle, Andriol could
have a role as a heavy cycle taper. There are also
indications that Andriol relieves depression in males
with normal testosterone levels. Of course, Andriol is an
expensive anti-depressant; St. John's Wort works for many
just as well and is cheaper.
2. Use for Taper
Even those who do not suffer from cycle termination
depression would find Andriol an effective, but
expensive, taper. For example, taper out of Sustanon with
primobo-depot and Andriol; reducing the primobo-d at a
rate such that the final taper element is low Andriol at
low dosage.
3. Use for Bridge
Another use for Andriol is as a 'bridge' between cycles.
In this respect it is perhaps more useful than 50mg deca-durabolin,
and certainly safer than testosterone enanthate. However,
in a bridging role Andriol (in common with other AS) will
not allow the recovery of the natural testosterone
production nor allow receptor recovery if taken at high
doses.
4. Use for Stack
Andriol can also be used as part of a stack of, for
example, deca-durabolin + primobo-depot and/or Anavar.
But in such cases Andriol should be viewed as a
supplement to, and not as the backbone of, the stack.
Here one would be seeking to benefit from the SHBG
suppression and synergistic effects referred to above.
Andriol can be stacked with any AS. WAR for example
suggests: Oxandrolone (p40, 225), deca-durabolin (p41, 84),
oral-turinabol (p217), and primobolan-depot (p240).
5. Use for Pre-Training
It is also suggested by some that Andriol should be used
as a pre-training supplement and, although there is no
consensus as to dose, it is often suggested that the
Andriol be taken 1 hour before a workout. There is no
clear evidence to support Andriol's role in this regard.
Given the nature of Andriol, it is doubtful whether
ingestion one hour prior to training would serve any
useful purpose.
More Effective Application?
Various suggestions have been made as to how Andriol
might be more effectively applied. These include (a)
extracting the TU from the capsule and injecting it, (b)
extracting the content of the capsules and applying it
topically with the aid of DMSO, (c) extracting the
content of the capsules and taking it in conjunction with
Vitamin E, (d) taking it with Saw Palmetto or Proscar,
and (e) taking it with grapefruit juice. There is no
evidence to show that any of these methods increases the
effectiveness of Andriol, but methods (d) and (e) do have
some logic to support them and may do some good. Indeed
for those BB concerned about their prostate and/or
potential hair loss, it is sensible to supplement any AS
cycle (Andriol or other) with Saw Palmetto. The proven
benefits of Saw Palmetto, especially for the older BB,
far outweigh the alleged marginal loss of 'gains' that
might arise from its use.
Cost
The current mail-order cost of Andriol from Europe varies
from $20 - $50 for 60 capsules. The pharmacy price of
Andriol in Europe varies from $14 for 60 capsules to $42
for 56 capsules. Andriol is not currently available from
pharmacies in the US.
Cautions
Although, Andriol is generally considered an almost
benign AS at low to moderate doses, caution is necessary
when taking it at high doses. Given the very
idiosyncratic nature of Andriol, it is impossible to be
precise as to what dose constitutes "high". WAR
implies that high is in the area of 240 - 280 mg/day (ie
6 - 7 capsules/day). At high doses, particularly if
sustained for an extended period, the normal BB using
Andriol will be exposed to the usual risks associated
with AS including suppression of the HPT axis, excess
estrogen problems, skin changes, hair loss, prostate
problems, etc.
The effectiveness of Andriol may be decreased even
further than outlined above, when some medicines are
taken in conjunction with it. The manufacturers specify
the following in this regard: antibiotics such as
rifampicin and anti-epileptic drugs such as barbitrates,
carbamazepine, dichloralphenazone, phenylbutazone,
phenytoin and primidone. Andriol will also potentiate the
effects of any anti-coagulants.
Those with allergies should know that Andriol contains a
form of sorbitol concentrate.
Anyone contemplating the use of Andriol should read the
excellent WAR section relating to it, and should also
consult the Rxmed website.
Conclusion
Andriol is a useful AS for the cautious BB, the older BB,
and the BB with medical problems. For the average BB it
is not cost effective, but if needs must, it can also be
utilised in an effective manner. It is perhaps
appropriate to point out that all BB will at some point
in their lives be older and/or cautious and/or medically
challenged. Thus all BB can, at some point in their
lives, utilise Andriol effectively.
Arimidex
Anastrozole [Oral]
Brand Names: Arimidex
Pronunciation: a-NAS-tro-zol
Drug class: Antineoplastic Agent
Generic available? No
Controlled substance? No
Oral anastrozole belongs to a class of antineoplastic
drugs called aromatase inhibitors. It is used as a second
phase treatment of breast cancer in postmenopausal women.
It works by decreasing estrogen levels in the body.
FDA Approved Uses
? Treatment of advanced breast cancer in post-menopausal
women with disease progression following tamoxifen
therapy.
Contraindications
Any of the
following may be reason to choose a different drug.
Inform your doctor before starting therapy.
? Hypersensitivity to anastrozole
Dosage and Administration
Dosages may
require modification to adjust for individual
sensitivities and associated medical conditions.
Adults Under 60
1 mg taken by mouth once per day.
Adults 60 and Over
Follow the adult dosage, unless directed otherwise by
your physician.
Maximum Dosage
Recommendations
Do not exceed the recommended doses, unless deemed
necessary by your doctor.
If You Miss a Dose
Take as soon as possible. If close to the next dose, skip
and take the next dose. Do not double the dose.
Storage
Keep all
medications out of the reach of children
Store in a tightly
closed container at room temperature in a dry, dark place.
Do not store in the bathroom. Moisture can cause the drug
to break down.
You may experience the following side effects with the
use of this drug:
Common Symptoms
? Dyspnea (shortness of breath)
? Dizziness
? Diarrhea
? Nausea or vomiting
? Headache
? Hot flashes
? Weakness
? Cough
? Dry mouth
? Skin rash
? Sweating
? Abdominal pain
? Bone pain
Less Common to Rare Symptoms
? Vaginal bleeding
? Weight gain
? Tiredness or weakness
? Cough or sore throat
? Muscle or joint pain
? Fever or chills
? Dizziness
? Breast pain
? Itching
Life-threatening Symptoms
? None expected
What to Do in Case of Overdose
Dial 911 for
emergency help or call your poison control center.
Prolonged Use
No problems are expected, providing you are not pregnant
when you start therapy, and do not become pregnant during
therapy.
Discontinuing
Therapy
Do not discontinue without your physician's consent
Back to top
Clenbuterol
This drug is classified as a beta-2 adrenergic agonist.
Clenbuterol is a bronchiodilator.This drug is banned by
the FDA although it is used outside the US by asthma
patients.The reason although it is fairly anabolic, and
it promotes the burning of fatty acids through brown fat
burning. Clenbuterol is a little scary because of some
other side effects including the following: tremors,
sweating, sleeplessness, rapid heartbeat, etc. These side
effects vary in people. Some people aren`t affected at
all. This drug comes in tablets of 20 mcg (micrograms not
milligrams ). Dosages are normally between 20-120 mcg for
bodybuilders that use this. It should be taken in a 2
days on /2days off fashion because this drug becomes
ineffective for its anabolic properties after 18
successive days of use. The receptor sites seem to be non-responsive
for anabolic purposes if taken continuously, but brown
fat-burning will continue past the 18 day period. It
shouldn`t be used this way for more than 12 weeks. After
12 weeks, the drug should be discontinued for a couple of
months.
Cheque
Drops
Cheque
drops are a veterinarian steroid made by Upjohn that is
designed to keep female dogs from going into heat. It
comes 100 mcg per cc, 55-cc bottle. It is the most toxic
androgenic steroid available. It is even more toxic than
say Finajet or Anadrol 50. Boxers and Powerlifters use it
to increase aggression and strength prior to training or
competition. It has been rumored that this is what caused
the infamous "ear-biting' incident that occurred
when Evander Holyfield last fought Mike Tyson. Users
report many side effects and little gains when using
Cheque Drops. It was very popular about 10 years ago but
has since faded away. It is very hard to obtain and is
not sought by many athletes. The drug itself is a
sublingual liquid that is dropped under the tongue and
gets in the system within a matter of minutes. The
athletes that were using this item would only take it
prior to a competition or prior to workouts and would not
use it any longer than two weeks at a time.
Clenbuterol
This
is a very interesting drug, which has recently become
popular amongst bodybuilders.
Clenbuterol itself, is a third generation beta agonist.
Clenbuterol's use as a bodybuilding drug item from a
number of medical reviews which have cited its
outstanding potential to promote muscle gains as well as
fat loss. It has been used in parts of England for
several years by a limited number of elite athletes. More
recently, due to the steroid crackdown, there have been
an increasing number of American bodybuilders that are
experimenting with this drug. Clenbuterol is indeed the
most intriguing ergogenic aid I have studied with the
sole exception of anabolic steroids.
Many athletes who use Clenbuterol claim that it promotes
dramatic strength increases and a very noticeable
reduction in body fat some athletes claim that they
enjoyed significant gains in muscle mass while using
Clenbuterol. Clenbuterol's most valid application seems
to be as a pre-contest, cutting drug. It is not banned by
any athletic committee; thus, numerous professional
bodybuilders have used it for the last month of contest
preparation. Athletes have used between 60-120 mcgs taken
in divided doses daily. Because it causes a great deal of
receptor downgrade it should not be used continually.
Research shows that using it for two days, then taking
two days off prevents attenuation. Cycles range from 6-12
weeks in length. Side effects include nervousness,
tremors of the hands, headaches, and insomnia. Usually
these side effects are dose related. It comes in 20 mcg
tablets. Clenbuterol is being counterfeited under
numerous manufacturer names in the United States.
Clomid
Clomid is a brand name for the drug clomiphene citrate.
It is typically prescribed for women to aid in ovulation.
In men, the application of Clomid causes an elevation of
follicle stimulating hormone and luteinizing hormone. As
a result, natural testosterone production is also
increased. This effect is obviously beneficial to the
athlete, especially at the conclusion of a cycle when
endogenous testosterone levels are subnormal. When an
athlete discontinues the use of steroids, his
testosterone levels will most likely be suppressed. If
endogenous testosterone levels are not brought to normal,
a dramatic loss in size and strength may occur. Clomid
plays a crucial role in preventing this crash in athletic
performance. Bodybuilders find that a daily intake of 50-100
mg of clomiphene citrate over a two week period will
bring endogenous testosterone production back to an
acceptable level. Clomid will gradually raise
testosterone levels over its period of intake. Since an
immediate boost in testosterone is often desirable,
athlete will commonly use HCG (human chorionic
gonadotropin) for a couple of weeks, and the continue
treatment with Clomid. Clomid is also effective as an
anti-estrogen. Most athletes will suffer from an elevated
estrogen level at the conclusion of a cycle. A high
estrogen level combined with a low testosterone level
puts an athlete in serious risk of developing
gynocomastia. With the intake of Clomid, the athlete gets
the dual effect of blocking out some of the effects of
estrogen, while also increasing endogenous testosterone
production. In relation to toxicity and side effects,
Clomid is considered a fairly safe drug. Bodybuilders
seldom experience any problems, but possible side effects
include hot flashes and temporary blurred vision.
Clomiphene citrate is widely available on the black
market. Until recently, it was relatively easy to get
through foreign mail order. However, since the DEA is
playing an active role in pursuing mail-order operations
catering to athletes, Clomid is becoming harder to obtain.
Current prices are between $2-$4 per 50 mg tab. Generics
such as Clomiphene citrate by Anfarm in Greece are
frequently seen on the black market and can be purchased
for about $1 a tablet.
Cyclofenil
Cyclofenil is another non-steroidal ancillary drug used
by athletes, similar to HCG and Clomid in action. This
drug is most commonly used to increase endogenous
testosterone levels after a cycle in an attempt to avoid
a hard crash while waiting for your hormone levels to
naturally balance. Similar to HCG and Clomid, cyclofenil
seems to quickly and effectively raise natural levels.
Anecdotally however, cyclofenil does has the reputation
of being the weaker of the three. Like Clomid, cyclofenil
may also act as an anti-estrogen, binding to estrogen
receptor sites and blocking out other estrogens. This is
especially helpful when natural testosterone levels are
suppressed and an excess of estrogen may be present upon
steroid termination. It should also be noted that some
athletes have experimented with using cyclofenil not as a
post-cycle ancillary drug, but alone and solely for it's
anabolic properties. However, anyone familiar with
anabolics would likely be disappointed with the results
cyclofenil would bring, as it is not an extremely strong
product, and certainly would not work as well as
anabolics. Here in the U.S., Fertodur from Mexico is
probably the most commonly imported cyclofenil product
although it is produced in many other countries.
Currently, fakes should not be a problem with this
product.
Cytadren
Cytadren, the U.S. brand name for the drug
aminoglutethimide, is an interesting drug (non-steroid),
first brought to our attention a few years ago by Dan
Duchaine. It is most popular among competitive athletes
who are drug tested, as this substance is currently not
banned or tested for. Cytadren inhibits the production of
androgens, estrogens and cortisone (and related) in the
body. Medically, this drug is used to treat Cushing's
syndrome, an condition in which the body overproduces
cortisone. For athletes with normal blood levels, a
little less cortisone could still be a good thing. While
androgens give your muscle cells a message to increase
protein synthesis, cortisone gives the exact opposite
message, to breakdown amino acids. Since Cytadren also
inhibits androgen production, it is always used by
athletes with some form of testosterone. Together with
even a relatively small dose, one could shift the ratio
of anabolic to catabolic hormones in favor of the former.
Cytadren also effectively inhibits estrogen production
and androgen to estrogen conversion. Research is bare as
to the best way for athletes to administer Cytadren, but
anecdotal evidence suggests that a schedule of 2 days on
and 2 days off is effective. One thing is for certain,
when used by healthy individuals as an anti-catabolic,
Cytadren cannot be taken daily. After a short period of
regular use, your body will react to the lowered
cortisone levels and release increased amounts of another
hormone, ACTH, in response. Increased ACTH will result in
your body resuming cortisone production, basically making
Cytadren useless. When used medically though, a moderate
amount of hydrocortisone is supplemented to avoid this
reaction. For athletes however, this would probably be a
counterproductive practice. Thus the 2 day on 2 day off
regime has been implemented in an attempt to delay or
avoid this response. As for the daily dosage, athletes
have experimented with anywhere from 1/2 a tablet to 3
tablets per day (250mg), 1 or 2 being most common.
Cytadren is not without it's side effects and warnings
which are numerous.To be very succinct, these include,
but are not limited to, the possibility of fatigue,
dizziness, sleep disorder, apathy, depression, nausea/vomiting,
stomach upset, thyroid dysfunction and liver disease.
Athletes also report that the reduced cortisone often
brings about more aches in your joints and an increased
susceptibility to injury. Currently Cytadren is
expensive, around $2 a tab, which is probably why it's
use has not become more wide spread.
Cytomel
Known Name Brands: Cynomel, Cyronine, Cytomel, Cytomel
Tabs, Euthroid,
Linomel, Liothyronin, Neo-Tiroimade, Ro-Thyronine, T3,
Tertroxin, Thybon,-forte
Thyrotardin, Ti-Tre, Tiromel, Tironina, Trijodthyronin,
Trijod.Sanabo,
Trijodthyr.50, Trijodthyr.Leo.
This product usually comes in bottles of 100 tablets at
25 mcgs each. It is available in a variety of doses
though ranging from 5 - 100 mcgs. per tablet. Cytomel is
a synthetic thyroid hormone (Type T-3). There are two
main types of synthetic thyroid hormones that are
available being this and Synthroid (T-4). This product is
regarded as the stronger of the two products (it is 4-5
times stronger than Synthroid). This product works by
increasing the synthesis of protein, carbohydrates, and
fats as well as RNA in the body thereby increasing your
BMR (Basal Metabolic Rate). Bodybuilders love this
product for many reasons. This product is an excellent
fat burner since your metabolism is greatly increased
while being on it. You can afford to be a little sloppier
on precontest dieting since it will still burn fat when
you are taking in a lot of calories since your metabolism
is going haywire. Step over Ripped Fuel, E/C/A stack,
Thermodrine. When taken with clenbuterol, this is the
single best fatburning combination that is available
today (with the possible exception of DNP). It also helps
to make steroids more effective since it is such a good
aid for protein synthesis.Most people need to be careful
to start with a low dosage, about 25 mcgs. per day and
increase by about one tab or 25 mcgs. per day every 5-6
days. Make sure that you don't go over 100 mcgs. per day
at the very most. On days that you take muliple tabs,
divide the tabs evenly across the day (i.e. 100 mcgs.
would be 4 doses of 25 mcgs. apiece spread evenly across
the day.) You also need to make sure that you cycle down
off this product as well to keep the thyroid functioning
properly as well. Don't take for more than 5 weeks at a
time as well. After doing a cycle of this drug, make sure
you go at least 8 weeks before doing it again as to allow
normal thyroid functioning to return.
Back to top
|