Dear friend and fellow athlete,
Boasting an astounding 50% increase
in metabolic rate, DNP is the most effective fat burner that bodybuilders
are using today to melt away the last amounts of diet resilient fat on
their physiques. For comparison purposes, the ECA stack, which is also
a highly effective fat loss tool, produces only a 3% increase in metabolic
rate. Athletes reporting fat losses of 10-12 pounds in 8 days of use
have further added to the DNP mystique. However, DNP is also the deadliest
substance used in bodybuilding – so deadly, that it has killed
athletes including one member of Elite Fitness.
In this issue of Elite Fitness News, I’ll tell you more about DNP,
share the precautions you should take if you decide to use it, and give
you the reasons why you should avoid it in favor of other diet drugs
and supplements that are not nearly so dangerous.
DNP or 2,4-Dinitrophenol, (Pronounced die ni'tro fe' nolz) is an industrial
chemical with various applications such as making dyes, wood preservatives,
explosives, insect control substances, other chemicals, and as a photographic
developer. Sold under several trade names, including Caswell No. 392,
Sulfo Black B, and Nitro Kleenup, DNP has recently gained steady popularity
as a fat loss tool.
DNP was used in diet pills in the 1930s, but was banned for this use
in 1938. Classified as an "uncoupler of oxidative phosphorylation," medically,
DNP is quite dangerous. You see, the body has no negative feedback system
that may deal with overdoses. Specifically, there is no upper limit to
the increase in body temperature that may be obtained with DNP’s
use.
The following article combines several theories to form what is perhaps
the single best way to cycle DNP for maximum fat-loss benefits. As I
mentioned earlier, DNP can be deadly and I would never use it myself
nor would I ever recommend that anyone ingest it. The casual use of DNP
for dieting is ridiculous. Hearing reports of athletes using DNP before
trying a Cyclical Ketogenic Diet, legal diet supplements, and medically
supervised weight loss drugs is crazy. Here are a few links to effective
weight loss supplements, drugs, and strategies that are much safer than
DNP and are certainly a much better alternative for all but the most
elite bodybuilders.
That said, if an athlete makes the personal decision to use DNP, it is
possible to take precautions to maximize its benefits and minimize the
potential risks.
The 7-day DNP fat loss inferno cycle:
The 7-day DNP fat loss inferno cycle involves a moderate to high dosage
of DNP for fat burning. The DNP fat loss inferno involves a 7-day on,
7-day off approach with four distinct phases. Most athletes using DNP
follow this type of cycle. The phases are as follows:
Phase 1: The 3-day Carb-Depletion Phase.
Phase 2: The 1-day Thyroxine (T3) Re-normalization Phase.
Phase 3: The 14-day DNP Inferno Phase.
Phase 4: The 2-day Post-DNP Phase.
Phase 1. The 3-day Carb-depletion phase
Phase One has a three-day duration and begins the four days preceding
the ingestion of DNP. The purpose of this phase is to deplete muscle-glycogen
content by restricting carbohydrates. This is achieved through a Ketogenic
style diet.
Kcals should be restricted to 10-12 times bodyweight in lbs. And carbohydrates
should be restricted to less than 60g/day. Protein is consumed at 1 gram
per pound of bodyweight or higher and the remaining dietary calories
should come from fat.
This phase lasts exactly 3 days, and will reduce muscle-glycogen levels
so that the body is forced to rely on fat as fuel more readily when you
start your DNP cycle.
Phase 2 The 1-day Thyroxine (T3) Re-normalization Phase
This is a new concept for DNP dieting. During the past three days, the
athlete has restricted carbohydrates and as a direct consequence T4-T3
conversion is slowed down resulting in reduced T3 levels. This is bad
for the DNP phase, as you need enough active T3 to last throughout the
entire 7-day on DNP phase.
Day four of the DNP cycle involves a mega-carbohydrate meal at mid-afternoon
(4-6PM) designed to create a massive insulin spike and re-normalize T4-T3.
This concept has been extrapolated from ketogenic diets and has been
shown to dramatically increase serum concentrations of T3.
Day 4 involves Keto eating until the Mega-carb meal. Then in the late
afternoon, at least circa 250g of carbohydrates must be consumed to create
an insulin spike. Any sugar (fructose, sucrose, maltose etc.) is fair
game. Fructose in particular is good because it primarily re-fills liver
glycogen which is directly involved in T4-T3 conversion. (Empty liver
glycogen signals the thyroid to decrease T4-T3 conversion).
As a side-note, a 250g carb-meal after three days of Keto dieting creates
a more pronounced insulin spike than would a 250g carb-meal after three
days of normal eating.
Kcals during Phase 2 should be kept at 15X Bodyweight in lbs. Macro-nutrient
break-downs can be calculated by the athlete. The only carb intake on
day 4 should be the 250g carb-meal.
Phase 3 The 14-Day DNP Phase
The first two days of actual DNP consumption are the most important to
follow correctly. During Days 1 and 2 of the actual DNP portion of the
cycle, it must be determined if the athlete will have an allergic reaction
to DNP.
Day 1: 200 mg of DNP is ingested
Day 2: 200 mg of DNP is ingested
At this point the dieter should be able to assess if an allergic reaction
has occurred. A DNP-stimulated allergic reaction will lead to swelling
in as little as 1 to 2 days time. Approximately 10% of athletes will
have such a reaction. The unfortunate few who experience this type of
a reaction must terminate the cycle immediately. Benadryl or Ketotifen
(Anti-histamines) can be used to treat mild symptoms. Obviously a doctor
should be consulted should the symptoms prove more severe.
Day 3: Dieters making it to day 3 of the DNP phase have the option of
increasing their dosage. The normal dosage for beginners is 400mg DNP/day.
Even an amount this small should provide outstanding results. A word
of caution. DO NOT TAKE MORE, if you are not experienced with DNP-use.
More advanced users may chose to go higher based on past experience.
The 400mg/day dosage is maintained from Day 3 through Day 9(Exactly 7
days). The last dose is taken on Day 9.
Supplementation and Nutritional Protocol for a DNP cycle:
1. An ECA stack is beneficial while on a DNP cycle as it as it acts as
an anorectant. DNP raises Neuro-peptide Y levels in the brain, which
is directly linked to increased hunger. Consuming 75-100mg total of ephedrine
alkaloids/day should be sufficient to suppress appetite. PPA (Nor-ephedrine)
should NOT be used as it causes lethargy when combined with DNP.
2. Anti-oxidants. Due to the DNP induced rapid combustion of fats, free-radical
production skyrockets up-wards. To combat this, anti-oxidants must be
used. Anti-oxidants are the single most important supplement to take
on a DNP cycle.
a) Fat-soluble Anti-O: Vitamin E: 1000mgs/day
b) Water-soluble Anti-O: Vitamin C: 2-3g/day
c) Alpha Lipoic acid: 600-1000mgs/day
Dual-anti-oxidant: BOTH fat & water-soluble actually re-cycles other
anti-oxidants.
3. Glycerol: Although optional, glycerol is often consumed at 15ml's
3X/day. Glycerol increases hydration for many athletes.
No additional supplements are really required other than these three.
All the rest you have read in various DNP articles are more for peace
of mind than improved functionality. I consider them overkill.
4. Water: Not a supplement, but an absolute necessity.
DNP causes sweating and can be incredibly dehydrating. Dehydration is
the NUMBER ONE cause of most DNP problems and deaths. Excessive dehydration
results in over-heating. Dieters who do not replenish fluids properly
while on a DNP cycle could die. The consensus among athletes is that
at least two gallons of water must be consumed daily.
5. EAT FRUIT while on your DNP cycle.
Fruit for some reason has been found to greatly reduce the lethargy associated
with a DNP cycle. It also has a high water content, therefore it helps
to keep the dieter hydrated. Watermelon is an obvious recommendation.
6. Dietary intake: There are several schools of thought on this matter,
but sticking to the old standard always works.
Kcals should be kept anywhere from 10-15X Bodyweight in lbs. Macro-nutrient
break-downs should be kept at around 20% fat, 30% protein and 50% carbs.
(Changing the ratios in favor of more carbs and protein w/ less fat will
result in a more fat loss but nothing special. Also, remember that more
carbohydrates means more heat.)
Take for example the 220 lb (100 kg) bodybuilder. He would consume anywhere
from 2200 to 3300Kcal /day (Depending on his appetite control).
WHAT NOT TO DO on a DNP cycle.
a) Do not under any circumstances consume alcohol or ANY type of diuretic
while on a DNP cycle. Alcohol and diuretics will dehydrate you and can
cause SERIOUS problems.
b) Do not remain in a hot environment without replenishing fluid loss
due to perspiration. This too can also cause SERIOUS problems.
c) Do not begin with a high dosage of DNP if you are a novice. This is
just asking for a trip to the ICU.
The half-life of 2,4 Dinitrophenol is 36 hours. So, after 36 hours, there
is only 50% of the DNP remaining in your system. Therefore, 72 hours
later 25% remains. Then 12.5% remains after 108 hours. After 5 days (120
hours), there's roughly 9% of the DNP left in your body that you had
on Day 9. This DNP concentration is low-enough to allow you to begin
Phase 4 of the cycle -- the 2-day Post-DNP phase -- without compromising
glycogen synthesis rates. Kcals during Days 10-14 should remain the same
as during days 3-9.
Phase 4: The 2 day Post DNP Phase.
The whole purpose of this phase is to get muscle-glycogen levels back
to normal. The Ketogenic carb-up can be used as a sort of template for
this phase.
After Phases two and three, muscle-glycogen levels are depressed and
need to be replenished.
Day 15: Carb-intake should be 7g/Kg of LBM (lean body mass = bodyweight
minus body fat.) So assuming a 220 lb bodybuilder has 0% body fat, lol,
he would consume 700 g of Carbs. Protein-intake remains at 1g/lb and
fat is restricted as low as possible.
The focus on day 1 should be on High-GI foods like Fat-free Ice-cream
and all the other non-fat high sugar desserts. Calories should be around
4000 for the 220-lb bodybuilder -- in other words, 18X bodyweight in
lbs.
Drastically restricting fat is CRITICAL here, as the body is still burning
fat for fuel as you replenish your glycogen stores. In essence, the dieter
is still losing fat while carbing up.
Day 16: Muscle-glycogen has increased, so carb-intake should be decreased
from day one’s 7g/Kg to only 5g/Kg of LBM. That would be 500g for
our 220-lb bodybuilder. Protein is 1g/lb again. Fat remains as low as
possible. Kcals for the dieter are reduced to 3000 Kcal range, or around
14X Bodyweight in lbs. The focus of Day 2 should be low-GI foods like
vegetables, milk, lean meats etc.
Additional Precautions:
Dieters feeling extremely nauseated or who vomit during a cycle should
discontinue use immediately and not restart for at least 36 hours.
Dieters should carry a pocket thermometer at all times. If body temperature
rises above 102 Fahrenheit then the dosage should be lowered or the cycles
should be terminated. Additionally, the dieter should take a very cold
bath to lower the temperature.
In addition to water, V8 juice should be consumed. Drinking gallons of
water depletes the body of electrolytes pretty badly predisposing the
dieter to shock, nausea, lethargy, and even death. V8 is the best for
replenishing electrolytes as it contains 950mg of potassium per 8oz compared
to Gatorade’s
35mg of potassium in 8oz.
Massive amounts of fruits and sweets should be consumed if one becomes
nauseated or vomits – i.e. force feed yourself.
Dieters should never allow themselves to become overheated on a DNP cycle.
Always stay next to a fan and keep the air conditioner on. Do not attempt
a DNP cycle if you work out doors in a warm climate or another warm environment
like a kitchen. Even at low doses this can build up and be potentially
dangerous.
There are two versions of DNP – regular and crystalline. Know
which one you are taking. When taking the crystalline DNP caps, never
take more than 200mg at once if you've never used it before. Even if
you are used to it, it is still much safer to spread the dosage throughout
the day. Crystalline DNP is much faster acting and can rapidly elevate
temperature.
Post-Steroid Cycle Use of DNP
One of the primary causes of muscle breakdown after a steroid cycle is
suppressed TSH. Anabolic steroids suppress TSH, which in turn lowers
T3 and T4 production by the thyroid gland. The reduction in TSH is one
reason that anabolic steroids are such excellent muscle builders.
Soon after the completion of a steroid cycle, TSH up-regulates, which
in turn super-stimulates the thyroid. This excess stimulation causes
the thyroid to produce above normal levels of T3 and T4. This increase
in thyroid hormones is highly catabolic and is the main reason why people
lose muscle post-cycle.
Athletes have learned that they need to restrict T3 production post cycle
to prevent muscle loss. A novel approach to achieving this goal is the
use of DNP. About 80% of the body’s endogenous T3 is produced from
the metabolically inactive T4 to the metabolically active T3. The de-iodinase
enzyme is responsible for this conversion. It literally cleaves off an
iodine molecule.
By ingesting 200mg DNP/day, the athlete can correct the over stimulated
Thyroid, returning T3 levels back to normal. DNP directly blocks the
production of T3 from T4 via the de-iodinase enzyme.
As a bonus, the reduction in your ATP stores because of the DNP is counter
acted by an increase in the oxidation of triglycerides as an energy source.
The benefit is the elimination of any potential fat-gain from the low
post-cycle testosterone levels. And as DNP is non-hormonal, it has no
effect on HPTA recovery.
After cessation of DNP use post-cycle, the athlete will reap the benefits
of the "Anabolic Rebound Effect" which further lends credence to the
use of DNP as a post-cycle ancillary for the elimination of any post-cycle
muscular losses.
Macro’s DNP Supplements
200mg alpha lipoic acid 3x a day with meals
1200-1500mg magnesium in 2-3 divided doses.
2-3000mg vitamin C
1200IU of vitamin E
200mcg of selenium.
1000-2000mg of calcium (can’t take it with the magnesium, though.
Take it before bed)
Melatonin if you can’t sleep and it is also one of the best and
cheapest anti-oxidants.
50mg of zinc a day
one iron tab as hemoglobin is a protein as well.
A potassium gluconate tab or two a day
Taurine at 3g a day.
Glutamine at 15g-20g a day .
1 table spoon glycerol 3 x a day
at least 2 gallons of water
a fan to point at your head while sleeping- or at work- basically anytime
you can point a fan at you
500mg grapeseed extract
300mg cranberry extract
600-900mg of green tea
a good mulit vitamin
EC+1g of tyrosine 3x per day and 20mg of yohimbine topically 2x per day-
for added energy and fat burning effects
Calorie Charts and Glycemic Index Lists can be found here:
http://www.elitefitness.com/articles/
And here's a link to discuss this article on the EliteFitness.com Discussion Forums.
Yours in sport,
George Spellwin
elitefitness.com
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